Basic Peptide Information

DICL ID
DICL_Pep_04069
Ion Channel
Neuronal acetylcholine receptor subunit alpha-9/alpha-10
Peptide Function
Antagonist
Gene Name
CHRNA9/CHRNA10

Activity Data (nM)

IC50
22.2 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
GCCSHPACSVNHPELC
Peptide UniProt Accession
UniParc
UPI0001874811
Peptide Synonyms/Alias
α-PeIA
Peptide Species
Conus pergrandis (Grand cone)
Peptide Name
Alpha-conotoxin PeIA
CAS Number
Not available

Experimental Conditions

pH
Not mention
Holding Potential (mV)
−80 mV
Temperature
21−24 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available